1-32. (canceled)
33. A composition comprising an oil-in-water emulsion comprising: (a) allantoin; (b) an emulsifier system comprising: (i) an acidic anionic polymer; and (ii) a nonionic emulsifier that is an ethoxylated ether or an ethoxylated ester whose carbon chain length ranges from 8 to 22 carbon atoms, wherein the pH of the composition is from about 3.0 to about 6.0.
34. The composition of claim 33 wherein the pH of the composition is from about 5.0 to about 6.0.
35. The composition of claim 33 wherein the acidic anionic polymer is carboxypolymethylene.
36. The composition of claim 33 further comprising a carbohydrate polymer selected from the group consisting of galactoarabinan, polygalactose, and polyarabinose.
37. The composition of claim 36 wherein the carbohydrate polymer is galactoarabinan.
38. The composition of claim 33 wherein the emulsifier system further comprises glyceryl stearate.
39. The composition of claim 33 further comprising at least one of: (a) an emollient component comprising at least one emollient selected from the group consisting of lanolin oil, cetyl alcohol, stearyl alcohol, and cod liver oil; (b) butylated hydroxytoluene; (c) a solvent component comprising at least one solvent selected from the group consisting of glycerin, propylene glycol, and butylene glycol; and (d) a preservative component comprising at least one preservative selected from the group consisting of methylparaben, propylparaben, and diazolidinyl urea.
40-81. (canceled)
The claims below are in addition to those above.
All refrences to claim(s) which appear below refer to the numbering after this setence.
1. A compound of the formula I,
wherein
R1 is unsubstituted or substituted alkyl, unsubstituted or substituted mono- or bicyclic aryl, unsubstituted or substituted mono- or bicyclic heterocyclyl, unsubstituted or substituted mono- or bicyclic cycloalkyl, unsubstituted or substituted mono- or bicyclic aryl-alkyl, unsubstituted or substituted mono- or bicyclic heterocyclyl-alkyl, unsubstituted or substituted mono- or bicyclic cycloalkyl-alkyl, unsubstituted or substituted alkenyl, substituted or unsubstituted alkynyl or acyl;
R2 is unsubstituted or substituted alkyl, unsubstituted or substituted mono- or bicyclic aryl, unsubstituted or substituted mono- or bicyclic heterocyclyl, unsubstituted or substituted mono- or bicyclic cycloalkyl, unsubstituted or substituted bicyclic aryl-alkyl, unsubstituted or substituted mono- or bicyclic heterocyclyl-alkyl, unsubstituted or substituted mono- or bicyclic cycloalkyl-alkyl, unsubstituted or substituted alkenyl, substituted or unsubstituted alkynyl; with the proviso that if R1 is one of the moieties mentioned in the definition of R1 other than acyl then R2 can also be unsubstituted or substituted monocyclic aryl-alkyl;
R3 is a moiety selected from the group consisting of moieties of the formulae
\u2003where in any of the moieties of the formulae given above under (a), (b), (c), (d), (e), (f) and (g) the asterisk (*) shows the bond binding the respective moiety R3 to the rest of the molecule in formula I,
Ra is unsubstituted or substituted alkyl, unsubstituted or substituted mono- or bicyclic aryl, unsubstituted or substituted mono- or bicyclic heterocyclyl, unsubstituted or substituted mono- or bicyclic cycloalkyl, unsubstituted or substituted mono- or bicyclic aryl-alkyl, unsubstituted or substituted mono- or bicyclic heterocyclyl-alkyl, unsubstituted or substituted mono- or bicyclic cycloalkyl-alkyl, acyl or hydrogen;
Rb and Rc are independently selected from the group consisting of unsubstituted or substituted alkyl, unsubstituted or substituted mono- or bicyclic aryl, unsubstituted or substituted mono- or bicyclic heterocyclyl, unsubstituted or substituted mono- or bicyclic cycloalkyl, unsubstituted or substituted bicyclic aryl-alkyl, unsubstituted or substituted mono- or bicyclic heterocyclyl-alkyl, unsubstituted or substituted mono- or bicyclic cycloalkyl-alkyl, acyl or hydrogen, with the proviso that not more than one of Rb and Rc is acyl, and with the proviso that if Rc is one of the mentioned moieties other than acyl then Rb can also be unsubstituted or substituted monocyclic aryl-alkyl; or Rb and Rc may form together a 3 to 7 membered nitrogen containing ring which can be unsubstituted or substituted;
Rd in a moiety of the formula (c) is unsubstituted or substituted alkyl, unsubstituted or substituted mono- or bicyclic aryl, unsubstituted or substituted mono- or bicyclic heterocyclyl, unsubstituted or substituted mono- or bicyclic cycloalkyl, unsubstituted or substituted mono- or bicyclic aryl-alkyl, unsubstituted or substituted mono- or bicyclic heterocyclyl-alkyl, unsubstituted or substituted mono- or bicyclic cycloalkyl-alkyl or acyl, or can have one of these meanings or can be \u2014N(Rb)(Rc) if m is 1 or 2;
Re is hydrogen, unsubstituted or substituted mono- or bicyclic aryl-alkyl, unsubstituted or substituted mono- or bicyclic cycloalkyl-alkyl or substituted or unsubstituted C1-C7-alkyl; and
Rf is substituted alkyl or unsubstituted or substituted mono- or bicyclic aryl, unsubstituted or substituted mono- or bicyclic heterocyclyl, unsubstituted or substituted mono- or bicyclic cycloalkyl, unsubstituted or substituted mono- or bicyclic aryl-alkyl, unsubstituted or substituted mono- or bicyclic heterocyclyl-alkyl, unsubstituted or substituted mono- or bicyclic cycloalkyl-alkyl;
m is 0, 1 or 2;
each of R4 and R5 is selected, independently from the other, from hydrogen, unsubstituted or substituted alkyl, hydroxy or esterified or etherified hydroxy;
and T is methylene, methylene mono-substituted by alkyl, carbonyl or thiocarbonyl;
or a salt thereof.
2. The compound of the formula I according to claim 1, wherein
R1 is acyl;
R2 is unsubstituted or substituted cycloalkyl or unsubstituted or substituted alkyl,
R3 is a moiety selected from the group consisting of moieties of the formulae
where in any of the moieties of the formulae given above under (a), (b), (c) and (f) the asterisk (*) shows the bond binding the respective moiety R3 to the rest of the molecule in formula I,
Ra is acyl or hydrogen;
Rb is unsubstituted or substituted alkyl, unsubstituted or substituted mono- or bicyclic aryl, unsubstituted or substituted mono- or bicyclic aryl-C1-C7alkyl or acyl;
Rc is hydroxy-C1-C7alkyl, C1-C7alkyloxy-C1-C7alkyl or preferably C3-C8-cycloalkyl, hydrogen or C1-C7-alkyl;
Rd is unsubstituted or substituted mono- or bicyclic aryl-C1-C7alkyl;
Re is hydrogen or C1-C7-alkyl; and
m is 2;
each of R4 and R5 is selected, independently from the other, from hydrogen, unsubstituted or substituted alkyl, hydroxy or esterified or etherified hydroxy;
and T is methylene, methylene mono-substituted by alkyl, carbonyl or thiocarbonyl;
or a pharmaceutically acceptable salt thereof.
3. The compound of the formula I according to claim 1, wherein
R1 is phenyl-, indolyl-, quinolyl- or 2,3-dihydro-benzo1,4dioxinyl-C1-C7-alkanoyl wherein the phenyl, indolyl, quinolyl or 2,3-dihydro-benzo1,4dioxinyl is substituted by halo, C1-C7-alkyloxy-C1-C7-alkyloxy, C1-C7-alkylene-O\u2014C1-C7-alkyl or C1-C7-alkyloxy-C1-C7-alkyloxy-C1-C7-alkyl and may further be substituted by one or more C1-C7-alkyl andor C1-C7-alkyloxy moieties;
R2 is C3-C8-cycloalkyl or C1-C7-alkyl;
R3 is a moiety selected from the group of moieties of the formulae
where in any of the moieties of the formulae given above under (a), (b), (c) and (f) the asterisk (*) shows the bond binding the respective moiety R3 to the rest of the molecule in formula I,
wherein
Ra is hydrogen or N-mono- or N,N-di-(C1-C7-alkyl, (unsubstituted or halo-substituted) phenyl or naphthyl, phenyl-C1-C7-alkyl, naphthyl-C1-C7-alkyl C3-C8-cycloalkyl-C1-C7-alkyl, heterocyclyl-C1-C7-alkyl, heterocyclyl andor C3-C8-cycloalkyl)-aminocarbonyl;
each of Rb and Rc is, independently of the other, is selected from hydrogen, C1-C7-alkyl, C3-C8-cycloalkyl-C1-C7-alkyl, C3-C8-cycloalkyl, unsubstituted or substituted aryl, naphthyl-C1-C7-alkyl, or acyl, unsubstituted or mono-, di- or tri-(halo, C1-C7-alkoxy, C1-C7-alkyloxy-C1-C7-alkyoxy, C1-C7-alkyloxy-C1-C7-alkyl andor C1-C7-alkyl)-substituted phenyl- or naphthyl-C1-C7-alkanoyl, (tetrahydrofuranyl or tetrahydropyranyl)-carbonyl or (tetrahydrofuranyl or tetrahydropyranyl)-C1-C7-alkyl-carbonyl, C1-C7-alkylsulfonyl or (unsubstituted or C1-C7-alkyl-, halo-lower alkyl-, halo, C1-C7-alkyloxy-, cyano-, C1-C7-alkanoyl- andor C1-C7-alkylsulfonyl-substituted) (phenyl- or naphthyl)-C1-C7-alkylsulfonyl,
in particular acyl is selected from
(a) unsubstituted or substituted mono- or bicyclic aryl-carbonyl, wherein the aryl moiety is selected from phenyl, indanyl, or 1,2,3,4-tetrahydronaphthyl which is unsubstituted, mono- or di-substituted by heterocyclyl, heterocyclyl-CH2, \u2014O\u2014-C1-C7-alkyl, \u2014O\u2014C1-C7-alkylene-O-alkyl andor halo, whereby the heterocyclyl moiety in each case is monocyclic 5- or 6-membered heterocyclyl, containing an N andor O atom;
(b) unsubstituted or substituted mono- or bicyclic heterocyclylcarbonyl, wherein the heterocyclyl moiety is selected from 5 to 11 membered ring systems which may be saturated, partially saturated or aromatic, and having 1 or 2 heteroatoms selected from O andor N, including pyrazinyl, isoxazolyl, pyrrolidin-2-onyl, tetrahydrofuranyl, tetrahydropyranyl, indolyl, 2,3-dihydro-benzo1,4dioxinyl, chromanyl, 2H-chromenyl, 3,4-dihydro-1H-quinolin-2-onyl, benzodisoxazolyl, 4,5,6,7-tetrahydro-benzodisoxazolyl, 3a,4,5,6,7,7a-hexahydro-benzoaisoxazolyl, 1,4,5,6,-tetrahydro-cyclopentapyrazolyl, or 3,4-dihydro-2H-benzob1,4dioxepinyl, whereby the heterocyclyl moiety is unsubstituted or is mono-substituted with phenyl, \u2014C1-C7-alkyl or C3-C8-cycloalkyl;
(c) unsubstituted or substituted mono or bicyclic cycloalkylcarbonyl wherein the cycloalkyl moiety is selected from C3, C4, C5, C6 and C7-cycloalkyl which may be unsubstituted or mono-substituted with O\u2014C1-C4-alkyl or hydroxy;
(d) unsubstituted or substituted alkylcarbonyl wherein the alkyl moiety is selected from branched or straight chain C1-C7-alkyl, whereby the alkyl moiety is mono-substituted with \u2014O\u2014C1-C7-alkyl, hydroxyl, C1-C7-alkanoylamino, unsubstituted or di-substituted phenyloxy, aminocarbonyl, N -mono- or N,N-di-substituted aminocarbonyl and C1-C7-alkyloxycarbonyl;
(e) unsubstituted or substituted mono or bicyclic aryl-C1-C7-alkylcarbonyl, wherein the alkyl moiety may be mono-substituted with unsubstituted phenyl, C1-C7-alkanoylamino, O\u2014C1-C4-alkyl or hydroxyl, and wherein the aryl moiety is selected from phenyl or naphthyl, which may be unsubstituted or substituted by \u2014O\u2014C1-C7-alkyl, halo-C1-C7-alkyl, substituted phenyl, C1-C7-alkanoylamino andor halo;
(f) unsubstituted or substituted mono- or bicyclic heterocyclyl-C1-C7-alkylcarbonyl, wherein the Heterocyclyl moiety is selected from 5 to 11 membered ring systems which may be saturated, partially saturated or aromatic, and having 1 or 2 heteroatoms selected from O andor N, whereby the heterocyclyl moiety is unsubstituted or is mono-substituted with unsubstituted phenyl, \u2014C1-C7-alkyl or C1-C7-alkanoyl;
(g) unsubstituted or substituted mono or bicyclic cycloalkyl-C1-C7-alkylcarbonyl, whereby the alkyl moiety may be mono-substituted, including on the carbon where the cycloalkyl moiety is attached, with \u2014C1-C4-alkyl or hydroxyl, and wherein the cycloalkyl moiety is selected from C3, C5 and C6-cycloalkyl, which may be unsubstituted or mono-substituted with amino, O\u2014C1-C4-alkyl or hydroxy;
(h) unsubstituted or substituted alkyloxycarbonyl, wherein the alkyl moiety is from branched or straight chain C1-C7-alkyl and which may be mono-substituted with by \u2014O\u2014C1-C7-alkyl, C1-C7-alkanoylamino and N-mono- or N,N-di-substituted aminocarbonyl;
(i) unsubstituted or substituted mono- or bicyclic aryl-oxycarbonyl, wherein the aryl moiety is selected from phenyl or naphthyl, which may be unsubstituted, mono-substituted with heterocyclyl or \u2014O\u2014C1-C7-alkyl, whereby the heterocyclyl moiety is monocyclic 5- or 6-membered heterocyclyl, containing an N andor O atom;
(j) unsubstituted or substituted mono- or bicyclic heterocyclyloxycarbonyl, wherein the heterocyclyl moiety is selected from 5 to 7 membered ring systems which may be saturated, partially saturated or aromatic, and having 1 or 2 heteroatoms selected from O andor N, in particular tetrahydrofuranyl or tetrahydropyranyl, wherein the heterocyclyl moiety is unsubstituted;
(k) unsubstituted or substituted mono- or bicyclic cycloalkyloxycarbonyl wherein the cycloalkyl moiety is selected from C6-cycloalkyl which is unsubstituted;
(l) unsubstituted or substituted mono- or bicyclic aryl-C1-C7-alkyloxycarbonyl, wherein the aryl moiety is selected from phenyl which is unsubstituted;
(m) unsubstituted or substituted mono- or bicyclic heterocyclyl-C1-C7-alkyloxycarbonyl, wherein the cycloalkyl moiety is selected from 5 to 7 membered ring systems which may be saturated, partially saturated or aromatic, and having 1 or 2 heteroatoms selected from O andor N, which is unsubstituted or is mono-substituted with \u2014C1-C7-alkyl or C1-C7-alkanoyl;
(n) unsubstituted or substituted mono- or bicyclic cycloalkyl-C1-C7-oxycarbonyl, such as cycloalkyl-CH2\u2014, wherein the cycloalkyl moiety is selected from C3 and C5-cycloalkyl, and may be unsubstituted or substituted with C1-C7-alkanoylamino,
(o) N-mono- or N,N-di-(unsubstituted or substituted mono- or bicyclic aryl, unsubstituted or substituted mono- or bicyclic cycloalkyl, unsubstituted or substituted mono- or bicyclic aryl-C1-C7-alkyl, unsubstituted or substituted mono- or bicyclic heterocyclyl-C1-C7-alkyl, unsubstituted or substituted mono- or bicyclic cycloalkyl-C1-C7-alkyl andor unsubstituted or substituted alkyl) -aminocarbonyl, whereby
the alkyl moiety of the unsubstituted or substituted alkyl aminocarbonyl is branched or straight chain C1-C7-alkyl which is unsubstituted;
the aryl moiety of the unsubstituted or substituted aryl aminocarbonyl is phenyl or naphthyl, which is unsubstituted,
the cycloalkyl moiety of the unsubstituted or substituted cycloalkyl aminocarbonyl is C3 or C6-cycloalkyl which is unsubstituted;
the aryl alkyl moiety of the unsubstituted or substituted aryl alkyl aminocarbonyl is aryl-CH2\u2014, aryl-CH2CH2\u2014, or aryl-CH(CH2CH3)\u2014, whereby the alkyl moiety may be mono-substituted with unsubstituted phenyl, and whereby the aryl moiety is phenyl, which is unsubstituted;
the heterocyclyl alkyl moiety of the unsubstituted or substituted heterocyclyl alkyl aminocarbonyl is heterocyclyl-CH2\u2014 whereby the heterocyclyl moiety is selected from 5 to 7 membered ring systems which may be aromatic, and having 1 or 2 heteroatoms selected from O andor N; which is unsubstituted;
the cycloalkyl alkyl moiety of the unsubstituted or substituted cycloalkyl alkyl aminocarbonyl is cycloalkyl-CH2\u2014, whereby the cycloalkyl moiety is selected from C6-cycloalkyl which is unsubstituted;
with the proviso that if Rc is hydrogen, C1-C7-alkyl, phenyl, naphthyl or naphthyl-C1-C7-alkyl, then
Rb can also be phenyl-C1-C7-alkyl;
Rd is unsubstituted or C1-C7-alkyl-, phenyl-, halo-lower alkyl-, halo, oxo-C1-C7-alkyl-, C1-C7-alkyloxy-, phenyl-C1-C7-alkoxy-, halo-C1-C7-alkyloxy-, phenoxy-, C1-C7-alkanoylamino-, cyano-, C1-C7-alkanoyl- andor C1-C7-alkylsulfonyl-substituted (phenyl- or naphthyl)-C1-C7-alkyl;
Re is hydrogen; and
m is 2;
each of R4 and R5 is hydrogen; and
T is carbonyl or methylene;
or a salt thereof.
4. The compound of the formula I according to claim 1, selected from the group of compounds consisting of:
N-((3S*,4S*)-4-{(3-Acetylamino-3-methyl-butyryl)-cyclopropyl-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-(3S*,4S*)-4-({Cyclopropyl-2-(2-oxo-pyrrolidin-1-yl)-acetyl-amino}-methyl)-pyrrolidin-3-ylmethyl-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-(3S*,4S*)-4-({2-(1-Acetylamino-cyclopentyl)-acetyl-cyclopropyl-amino}-methyl)-pyrrolidin-3-ylmethyl-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S*,4S*)-4-{Cyclopropyl-(3,3-dimethyl-butyryl)-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-(3S*,4S*)-4-({2-(1-Acetylamino-cyclohexyl)-acetyl-cyclopropyl-amino}-methyl)-pyrrolidin-3-ylmethyl-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S*,4S*)-4-{Cyclopropyl-(3-methyl-3-pyrrol-1-yl-butyryl)-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-(3S*,4S*)-4-({Cyclopropyl-2-(3-oxo-3,4-dihydro-2H-benzo1,4oxazin-6-yl)-acetyl-amino}-methyl)-pyrrolidin-3-ylmethyl-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-(3S*,4S*)-4-({Cyclopropyl-2-(1-isobutyrylamino-cyclopentyl)-acetyl-amino}-methyl) -pyrrolidin-3-ylmethyl-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S*,4S*)-4-{Cyclopropyl-(4-methyl-pentanoyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-(3S*,4S*)-4-({Cyclopropyl-2-(2-methyl-benzooxazol-5-yl)-acetyl-amino}-methyl)-pyrrolidin-3-ylmethyl-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S*,4S*)-4-{(3-Cyclohexyl-propionyl)-cyclopropyl-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S,4S)-4-{Cyclopropyl-(3-cyclopropyl-propionyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S,4S)-4-{(3-Cyclopentyl-propionyl)-cyclopropyl-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S,4S)-4-{Cyclopropyl-(3,3-diphenyl-propionyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-(3S,4S)-4-({Cyclopropyl-2-(2,6-dimethyl-phenoxy)-acetyl-amino}-methyl)-pyrrolidin-3-ylmethyl-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S,4S)-4-{Cyclopropyl-((S)-3-phenyl-butyryl)-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-(3S,4S)-4-((2-(1-Acetyl-piperidin-4-yl)-acetyl-cyclopropyl-amino}-methyl)-pyrrolidin-3-ylmethyl-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S,4S)-4-{((S)-3-Acetylamino-3-phenyl-propionyl)-cyclopropyl-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S,4S)-4-{((R)-3-Acetylamino-3-phenyl-propionyl)cyclopropyl-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S,4S)-4-{Cyclopropyl-((R)-3-hydroxy-3-phenyl-propionyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S,4S)-4-{Cyclopropyl-((S)-3-hydroxy-3-phenyl-propionyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S,4S)-4-{Cyclopropyl-(3-furan-2-yl-propionyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S,4S)-4-{Cyclopropyl-(2-furan-2-yl-acetyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S,4S)-4-{Cyclopropyl-((S)-2-methoxy-2-cyclohexyl-acetyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S,4S)-4-{Cyclopropyl-((S)-2-hydroxy-4-methyl-pentanoyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-{(3S*,4S*)-4-(Cyclohexanecarbonyl-cyclopropyl-amino)-methyl-pyrrolidin-3-ylmethyl}-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
Cycloheptanecarboxylic acid cyclopropyl-(3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-amide
N-((3S,4S)-4-{(2-Cyclopentyl-acetyl)-cyclopropyl-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S*,4S*)-4-{(2-Cyclohexyl-acetyl)-cyclopropyl-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-{(3S*,4S*)-4-(Benzoyl-cyclopropyl-amino)-methyl-pyrrolidin-3-ylmethyl}-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-(3S*,4S*)-4-({Cyclopropyl-2-4-fluoro-phenyl)-acetyl-amino}-methyl)-pyrrolidin-3-ylmethyl-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-(3S,4S)-4-({2-(4-Chloro-phenyl)-acetyl-cyclopropyl-amino}-methyl)-pyrrolidin-3-ylmethyl-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-(3S*,4S*)-4-({2-(3-Chloro-phenyl)-acetyl-cyclopropyl-amino}-methyl)-pyrrolidin-3-ylmethyl-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-(3S*,4S*)-4-({Cyclopropyl-2-(2-methoxy-phenyl)-acetyl-amino}-methyl)-pyrrolidin-3-ylmethyl-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-(3S*,4S*)-4-({Cyclopropyl-2-(3,5-difluoro-phenyl)-acetyl-amino}-methyl)-pyrrolidin-3ylmethyl-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-(3S*,4S*)-4-({Cyclopropyl-2-2,3,5-trifluoro-phenyl)-acetyl-amino}-methyl)-pyrrolidin-3-ylmethyl-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-(3S*,4S*)-4-({Cyclopropyl-2-(3-trifluoromethyl-phenyl)-acetyl-amino}-methyl)-pyrrolidin-3-ylmethyl-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-(3S*,4S*)-4-{Cyclopropyl-(3-pyrrolidin-1yl-benzoyl)-amino-methyl}-pyrrolidin-3-ylmethyl-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-(3S*,4S*)-4-({Cyclopropyl-2-(3\u2032-fluoro-biphenyl-3-yl)-acetyl-amino}-methyl)-pyrrolidin-3-ylmethyl-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S*,4S*)-4-{Cyclopropyl-(3-chloro-6-methoxy-1-yl-benzoyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S*,4S*)-4-{Cyclopropyl-(4-morpholin-4-ylmethyl-benzoyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
1H-Indole-2-carboxylic acid cyclopropyl-(3S*,4S*)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-amide
1H-Indole-3-carboxylic acid cyclopropyl-(3S*,4S*)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-amide
2,3-Dihydro-benzo1,4dioxine-6-carboxylic acid cyclopropyl-(3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-amide
N-((3S*,4S*)-4-{Cyclopropyl-(2-naphthalen-2-yl-acetyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S,4S)-4-{Cyclopropyl-(2-phenoxy-acetyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S*,4S*)-4-{Cyclopropyl-((S)-2-phenyl-propionyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S*,4S*)-4-(Cyclopropyl-((R)-2-phenyl-propionyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S,4S)-4-{Cyclopropyl-((S)-2-hydroxy-2-phenyl-acetyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S,4S)-4-{Cyclopropyl-((R)-2-hydroxy-2-phenyl-acetyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S,4S)-4-{Cyclopropyl-((R)-2-methoxy-2-phenyl-acetyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S,4S)-4-{Cyclopropyl-((S)-2-methoxy-2-phenyl-acetyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
Tetrahydro-furan-3-carboxylic acid cyclopropyl-(3S*,4S*)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-amide
Tetrahydro-furan-2-carboxylic acid cyclopropyl-(3S*,4S*)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-amide
(S)-Tetrahydro-pyran-3-carboxylic acid cyclopropyl-(3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-amide
(R)-Tetrahydro-pyran-3-carboxylic acid cyclopropyl-(3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-amide
Tetrahydro-pyran-4-carboxylic acid cyclopropyl-(3S*,4S*)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-amide
N-((3S,4S)-4-{Cyclopropyl-(4-hydroxy-cyclohexanecarbonyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S,4S)-4-{Cyclopropyl-(cis-4-methoxy-cyclohexanecarbonyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S,4S)-4-Cyclopropyl-(trans-4-methoxy-cyclohexanecarbonyl)amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S,4S)-4-{Cyclopropyl-((S)-2-tetrahydro-furan-2-yl-acetyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S,4S)-4-{Cyclopropyl-((R)-2-tetrahydro-furan-2-yl-acetyl)-amino-methyl)-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S,4S)-4-{Cyclopropyl-((S)-2-tetrahydro-pyran-2-yl-acetyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-{3-methoxy-propoxy)-benzamide
N-((3S,4S)-4-{Cyclopropyl-((R)-2-tetrahydro-pyran-2-yl-acetyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
(R)-1,2,3,4-Tetrahydro-naphthalene-2-carboxylic acid cyclopropyl-(3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-amide
(S)-1,2,3,4-Tetrahydro-naphthalene-2-carboxylic acid cyclopropyl-(3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-amide
N-((3S*,4S*)-4-{Cyclopropyl-(2-tetrahydro-pyran-4-yl-acetyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
Chroman-2-carboxylic acid cyclopropyl-(3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-amide
2H-Chromene-3-carboxylic acid cyclopropyl-(3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-amide
(R)-2,3-Dihydro-benzo1,4dioxine-2-carboxylic acid cyclopropyl-(3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-amide
(S)-2,3-Dihydro-benzo1,4dioxine-2-carboxylic acid cyclopropyl-(3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-amide
2-Oxo-1,2,3,4-tetrahydro-quinoline-4-carboxylic acid cyclopropyl-(3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-amide
4,5,6,7-Tetrahydro-benzodisoxazole-3-carboxylic acid cyclopropyl-(3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-amide
3a,4,5,6,7,7a-Hexahydro-benzodisoxazole-3-carboxylic acid cyclopropyl-(3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-amide
N-((3S,4S)-4-{(2-Benzodisoxazol-3-yl-acetyl)-cyclopropyl-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
1,4,5,6-Tetrahydro-cyclopentapyrazole-3-carboxylic acid cyclopropyl-(3S*,4S*)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-amide
Isoxazole-3-carboxylic acid cyclopropyl-(3S*,4S*)-4-((isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-amide
5-Methyl-isoxazole-3-carboxylic acid cyclopropyl-(3S*,4S*)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-amide
5-Cyclopropyl-isoxazole-3-carboxylic acid cyclopropyl-(3S*,4S*)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-amide
5-Phenyl-isoxazole-3-carboxylic acid cyclopropyl-(3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-amide
5-Methyl-pyrazine-2-carboxylic acid cyclopropyl-(3S*,4S*)-4-({isopropyl-4methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-amide
Indan-2-carboxylic acid cyclopropyl-(3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-amide
5-Oxo-1-phenyl-pyrrolidine-3-carboxylic acid cyclopropyl-(3S*,4S*)-4-((isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-amide
N-Cyclopropyl-N-(3S*,4S*)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-succinamide
N-Cyclopropyl-N-(3S*,4S*)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-N\u2032-methyl-succinamide
N-Cyclopropyl-N-(3S*,4S*)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-succinamic acid methyl ester
N-((3S,4S)-4-{Cyclopropyl-(2-piperidin-4-yl-acetyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-(3S,4S)-4-({2-(4-Amino-cyclohexyl)-acetyl-cyclopropyl-amino}-methyl)-pyrrolidin-3-ylmethyl-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-(3S,4S)-4-({2-(4-Amino-cyclohexyl)-acetyl-cyclopropyl-amino}-methyl)-pyrrolidin-3-ylmethyl-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S,4S)-4-{Cyclopropyl-(2-methyl-2-phenyl-propionyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S,4S)-4-{((S)-2-Hydroxy-2-phenyl-acetyl)-methyl-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S,4S)-4-{((S)-2-Methoxy-2-phenyl-acetyl)-methyl-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S,4S)-4-{((S)-2-Hydroxy-4-methyl-pentanoyl)-methyl-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S,4S)-4-{((S)-2-Methoxy-2-cyclohexyl-acetyl)-methyl-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S,4S)-4-{((S)-2-Hydroxy-3-methyl-butyryl)-methyl-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S,4S)-4-{((S)-2-Hydroxy-3-phenyl-propionyl)-methyl-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S,4S)-4-(((S)-2-Cyclohexyl-2-hydroxy-acetyl)-methyl-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S ,4S)-4-{((S)-3-Hydroxy-3-phenyl-propionyl)-methyl-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S,4S)-4-{((R)-3-Hydroxy-3-phenyl-propionyl)-methyl-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S,4S)-4-{(2-Furan-2-yl-acetyl)-methyl-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S,4S)-4-{((S)-2-Methoxy-3-methyl-butyryl)-methyl-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S,4S)-4-{((S)-2-Methoxy-4-methyl-pentanoyl)-methyl-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S*,4S*)-4-(Benzoyl-methyl-amino)-methyl-pyrrolidin-3-ylmethyl}-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S,4)-4-{(2-Cyclohexyl-acetyl)-methyl-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3methoxy-propoxy)-benzamide
N-Isopropyl-4-methoxy-N-(3S*,4S*)-4-({2-(3-methoxy-phenyl)-acetyl-methyl-amino}-methyl)-pyrrolidin-3-ylmethyl-3-(3-methoxy-propoxy)-benzamide
Indan-2-carboxylic acid (3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-methyl-amide
(R)-1,2,3,4-Tetrahydro-naphthalene-2-carboxylic acid (3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-methyl-amide
(S)-1,2,3,4-Tetrahydro-naphthalene-2-carboxylic acid (3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-methyl-amide
Tetrahydro-pyran-4-carboxylic acid (3S*,4S*)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-methyl-amide
N-(3S,4S)-4-({2-(1-Hydroxy-cyclohexyl)-acetyl-methyl-amino}-methyl)-pyrrolidin-3-ylmethyl-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-Isopropyl-4-methoxy-N-(3S,4S)-4-({2-(4-methoxy-cyclohexyl)-acetyl-methyl-amino}-methyl)-pyrrolidin-3-ylmethyl-3-(3-methoxy-propoxy)-benzamide
N-Isopropyl-4-methoxy-N-(3S,4S)-4-({2-(4-methoxy-cyclohexyl)-acetyl-methyl-amino}-methyl)-pyrrolidin-3-ylmethyl-3-(3-methoxy-propoxy)-benzamide
3,4-Dihydro-2H-benzob1,4dioxepine-2-carboxylic acid (3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-methyl-amide
N-Isopropyl-4-methoxy-N-((3S,4S)-4-{(cis-4-methoxy-cyclohexanecarbonyl)-methyl-amino-methyl}-pyrrolidin-3-ylmethyl)-3-(3-methoxy-propoxy)-benzamide
N-Isopropyl-4-methoxy-N-((3S,4S)-4-{(trans-4-methoxy-cyclohexanecarbonyl)-methyl-amino-methyl}-pyrrolidin-3-ylmethyl)-3-(3-methoxy-propoxy)-benzamide
N-Isopropyl-4-methoxy-3-(3-methoxy-propoxy)-N-(3S,4S)-4-(phenylacetylamino-methyl)-pyrrolidin-3-ylmethyl-benzamide
Indan-2-carboxylic acid (3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-amide
N-{(3S,4S)-4-((S)-2-Cyclohexyl-2-methoxy-acetylamino)-methyl-pyrrolidin-3-ylmethyl}-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-Isopropyl-4-methoxy-N-{(3S,4S)-4-((R)-2-methoxy-2-phenyl-acetylamino)-methyl-pyrrolidin-3-ylmethyl}-3-(3-methoxy-propoxy)-benzamide
N-Isopropyl-4-methoxy-N-{(3S,4S)-4-((S)-2-methoxy-2-phenyl-acetylamino)-methyl-pyrrolidin-3-ylmethyl}-3-(3-methoxy-propoxy)-benzamide
N-{(3S,4S)-4-((R)-2-Cyclohexyl-2-methoxy-acetylamino)-methyl-pyrrolidin-3-yl methyl}-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-{(3S,4S)-4-(Ethyl-phenylacetyl-amino)-methyl-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S,4S)-4-{Ethyl-(2-tetrahydro-pyran-4-yl-acetyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-{(3S*,4S*)-4-(Cyclobutyl-phenylacetyl-amino)-methyl-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S*,4S*)-4-Cyclobutyl-(2-tetrahydro-pyran-4-yl-acetyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-Isopropyl-N-{(3S*,4S*)-4-(isopropyl-phenylacetyl-amino)-methyl-pyrrolidin-3-ylmethyl}-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-Isopropyl-N-((3S*,4S*)-4-{isopropyl-(2-tetrahydro-pyran-4-yl-acetyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-{(3S*,4S*)-4-(Cyclopropanecarbonyl-isobutyl-amino)-methyl-pyrrolidin-3-ylmethyl}-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S*,4S*)-4-(Cyclobutanecarbonyl-isobutyl-amino)-methyl-pyrrolidin-3-ylmethyl}-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S*,4S*)4-{Isobutyl-(2-tetrahydro-pyran-4-yl-acetyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-{(3S*,4S*)-4-(Isobutyl-phenylacetyl-amino)-methyl-pyrrolidin-3-ylmethyl}-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-{(3S*,4S*)-4-(Cyclopropylmethyl-phenylacetyl-amino)-methyl-pyrrolidin-3-ylmethyl}-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-((3S*,4S*)-4-{Cyclopropylmethyl-(2-tetrahydro-pyran-4-yl-acetyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
1-(3-Methoxy-propyl)-3-methyl-1H-indole-6-carboxylic acid isopropyl-{(3S,4S)-4-(methyl-phenylacetyl-amino)-methyl-pyrrolidin-3-ylmethyl}-amide
1-(3-Methoxy-propyl)-3-methyl-1H-indole-6-carboxylic acid ((3S,4S)-4-{(2-cyclohexyl-acetyl)-methyl-amino-methyl}-pyrrolidin-3-ylmethyl)-isopropyl-amide
N-{(3S,4S)-4-(Cyclopropyl-phenylacetyl-amino)-methyl-pyrrolidin-3-ylmethyl}-4-ethyl-N-isopropyl-3-(3-methoxy-propoxy)-benzamide
N-((3S,4S)-4-{(2-Cyclohexyl-acetyl)-methyl-amino-methyl}-pyrrolidin-3-ylmethyl)-4-ethyl-N-isopropyl-3-(3-methoxy-propoxy)-benzamide
4-Ethyl-N-isopropyl-3-(3-methoxy-propoxy)-N-((3S,4S)-4-{methyl-(2-tetrahydro-pyran-4-yl-acetyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-benzamide
Tetrahydro-pyran-4-carboxylic acid (3S,4S)-4-({4-ethyl-3-(3-methoxy-propoxy)-benzoyl-isopropyl-amino}-methyl)-pyrrolidin-3-ylmethyl-methyl-amide
N-((3S,4S)-4-{Cyclopropyl-(2-tetrahydro-pyran-4-yl-acetyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-4-ethyl-N-isopropyl-3-(3-methoxy-propoxy)-benzamide
Tetrahydro-pyran-4-carboxylic acid cyclopropyl-(3S,4S)-4-({4-ethyl-3-(3-methoxy-propoxy)-benzoyl-isopropyl-amino}-methyl)-pyrrolidin-3-ylmethyl-amide
N-((3S,4S)-4-{(3-Acetylamino-3-methyl-butyryl)-cyclopropyl-amino-methyl}-pyrrolidin-3-ylmethyl)-4-ethyl-N-isopropyl-3-(3-methoxy-propoxy)-benzamide
4-Ethyl-N-((3S,4S)-4-{((S)-2-hydroxy-2-phenyl-acetyl)-methyl-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-3-(3-methoxy-propoxy)-benzamide
N-(3S,4S)-4-({2-(1-Acetyl-piperidin-4-yl)-acetyl-cyclopropyl-amino}-methyl)-pyrrolidin-3-ylmethyl-4-ethyl-N-isopropyl-3-(3-methoxy-propoxy)-benzamide
N-(3S,4S)-4-({2-(1-Acetyl-piperidin-4-yl)-acetyl-methyl-amino}-methyl)-pyrrolidin-3-ylmethyl-4-ethyl-N-isopropyl-3-(3-methoxy-propoxy)-benzamide
4-Ethyl-N-((3S,4S)-4-{((S)-2-hydroxy-4-methyl-pentanoyl)-methyl-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-3-(3-methoxy-propoxy)-benzamide
4-Ethyl-N-((3S,4S)-4-{((S)-2-hydroxy-3-methyl-butyryl)-methyl-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-3-(3-methoxy-propoxy)-benzamide
Indan-2-carboxylic acid (3S,4S)-4-({4-ethyl-3-(3-methoxy-propoxy)-benzoyl-isopropyl-amino}-methyl)-pyrrolidin-3-ylmethyl-amide
4-Ethyl-N-isopropyl-3-(3-methoxy-propoxy)-N-{(3S,4S)-4-(2-methyl-2-phenyl-propionylamino)-methyl-pyrrolidin-3-ylmethyl}-benzamide
4-Ethyl-N-isopropyl-N-{(3S,4S)-4-((R)-2-methoxy-2-phenyl-acetylamino)-methyl-pyrrolidin-3-ylmethyl}-3-(3-methoxy-propoxy)-benzamide
N-(3S,4S)-4-({2-(4-Amino-cyclohexyl)-acetyl-methyl-amino}-methyl)-pyrrolidin-3-ylmethyl-4-ethyl-N-isopropyl-3-(3-methoxy-propoxy)-benzamide
N-(3S,4S)-4-({2-(4-Amino-cyclohexyl)-acetyl-methyl-amino}-methyl)-pyrrolidin-3-ylmethyl-4-ethyl-N-isopropyl-3-(3-methoxy-propoxy)-benzamide
5-Methyl-pyrazine-2-carboxylic acid (3S,4S)-4-({4-ethyl-3-(3-methoxy-propoxy)-benzoyl-isopropyl-amino}-methyl)-pyrrolidin-3-ylmethyl-methyl-amide
(S)-2,3-Dihydro-benzo1,4dioxine-2-carboxylic acid (3S,4S)-4-({4-ethyl-3-(3-methoxy-propoxy)-benzoyl-isopropyl-amino}-methyl)-pyrrolidin-3-ylmethyl-methyl-amide
(R)-2-Oxo-1,2,3,4-tetrahydro-quinoline-4-carboxylic acid (3S,4S)-4-({4-ethyl-3-(3-methoxy-propoxy)-benzoyl-isopropyl-amino}-methyl)-pyrrolidin-3-ylmethyl-methyl-amide
(S)-2-Oxo-1,2,3,4-tetrahydro-quinoline-4-carboxylic acid (3S,4S)-4-({4-ethyl-3-(3-methoxy-propoxy)-benzoyl-isopropyl-amino}-methyl)-pyrrolidin-3-ylmethyl-methyl-amide
N-Cyclopropyl-N-(3S,4S)-4-({4-ethyl-3-(3-methoxy-propoxy)-benzoyl-isopropyl-amino}-methyl)-pyrrolidin-3-ylmethyl-N\u2032-methyl-succinamide
5-Methyl-pyrazine-2-carboxylic acid cyclopropyl-(3S,4S)-4-({4-ethyl-3-(3-methoxy-propoxy)-benzoyl-isopropyl-amino}-methyl)-pyrrolidin-3-ylmethyl-amide
Isoxazole3-carboxylic acid cyclopropyl-(3S,4S)-4-({4-ethyl-3-(3-methoxy-propoxy)-benzoyl-isopropyl-amino}-methyl)-pyrrolidin-3-ylmethyl-amide
N-(3S,4S)-4-({2-(4-Amino-cyclohexyl)-acetyl-cyclopropyl-amino}-methyl)-pyrrolidin-3-ylmethyl-4-ethyl-N-isopropyl-3-(3-methoxy-propoxy)-benzamide
N-(3S,4S)-4-({2-(4-Amino-cyclohexyl)-acetyl-cyclopropyl-amino}-methyl)-pyrrolidin-3-ylmethyl-4-ethyl-N-isopropyl-3-(3-methoxy-propoxy)-benzamide
(R)-Tetrahydro-furan-3-carboxylic acid cyclopropyl-(3S,4S)-4-({4-ethyl-3-(3-methoxy-proxy)-benzoyl-isopropyl-amino}-methyl)-pyrrolidin-3-ylmethyl-amide
(S)-Tetrahydro-furan-3-carboxylic acid cyclopropyl-(3S,4S)-4-({4-ethyl-3-(3-methoxy-propoxy)-benzoyl-1-isopropyl-amino}-methyl)-pyrrolidin-3-ylmethyl-amide
(R)-Tetrahydro-pyran-3-carboxylic acid cyclopropyl-(3S,4S)-4-({4-ethyl-3-(3-methoxy-proxy)-benzoyl-isopropyl-amino}-methyl)-pyrrolidin-3-ylmethyl-amide
(S)-Tetrahydro-pyran-3-carboxylic acid cyclopropyl-(3S,4S)-4-({4-ethyl-3-(3-methoxy-propoxy)-benzoyl-isopropyl-amino}-methyl)-pyrrolidin-3-ylmethyl-amide
N-((3S,4 S)-4-{Cyclopropyl-(cis-4-hydroxy-cyclohexanecarbonyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-4-ethyl-N-isopropyl-3-(3-methoxy-propoxy)-benzamide
N-((3S,4S)-4-{Cyclopropyl-(trans-4-hydroxy-cyclohexanecarbonyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-4-ethyl-N-isopropyl-3-(3-methoxy-propoxy)-benzamide
(S)-Tetrahydro-pyran-3-carboxylic acid (3S,4S)-4-({4-ethyl-3-(3-methoxy-propoxy)-benzoyl-isopropyl-amino}-methyl)-pyrrolidin-3-ylmethyl-methyl-amide
(R)-Tetrahydro-pyran-3-carboxylic acid (3S,4S)-4-({4-ethyl-3-(3-methoxy-propoxy)-benzoyl-isopropyl-amino}-methyl)-pyrrolidin-3-ylmethyl-methyl-amide
N-Isopropyl-3-(3-methoxy-propoxy)-4-methyl-N-{(3S,4S)-4-(methyl-phenylacetyl-amino)-methyl-pyrrolidin-3-ylmethyl}-benzamide
Tetrahydro-pyran-4-carboxylic acid (3S,4S)-4-({isopropyl-3-(3-methoxy-propoxy)-4-methyl-benzoyl-amino}-methyl)-pyrrolidin-3-yl methyl-methyl-amide
N-Isopropyl-3-(3-methoxy-propoxy)-4-methyl-N-((3S,4S)-4-{methyl-(2-tetrahydro-pyran-4-yl-acetyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-benzamide
N-((3S,4S)-4-{Cyclopropyl-((S)-2-methoxy-2-phenyl-acetyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-3-(3-methoxy-propoxy)-4-methyl-benzamide
(S)-2,3-Dihydro-benzo1,4dioxine-2-carboxylic acid cyclopropyl-(3S,4S)-4-({isopropyl-3-(3-methoxy-propoxy)-4-methyl-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-amide
N-((3S,4S)-4-{((S)-2-Methoxy-2-phenyl-acetyl)-methyl-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-3-(3-methoxy-propoxy)-4-methyl-benzamide
(S)-2,3-Dihydro-benzo1,4dioxine-2-carboxylic acid (3S,4S)-4-({isopropyl-3-(3-methoxy-propoxy)-4-methyl-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-methyl-amide
N-((3S,4S)-4-{(3-Acetylamino-3-methyl-butyryl)-cyclopropyl-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-3-(3-methoxy-propoxy)-4-methyl-benzamide
N-((3S,4S)-4-{((S)-2-Hydroxy-2-phenyl-acetyl)-methyl-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-3-(3-methoxy-propoxy)-4-methyl-benzamide
Tetrahydro-pyran-4-carboxylic acid cyclopropyl-(3S,4S)-4-({isopropyl-3-(3-methoxy-propoxy)-4-methyl-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-amide
N-Isopropyl-3-(3-methoxy-propoxy)-4-methyl-N-(3S ,4S)-4-({methyl-2-(3-oxo-3,4-dihydro-2H-benzo1,4oxazin-6-yl)-acetyl-aminomethyl)-pyrrolidin-3-yl methyl-benzamide
N-(3S,4S)-4-({Cyclopropyl-2-(3-oxo-3,4-dihydro-2H-benzo1,4oxazin-6-yl)-acetyl-amino}-methyl)-pyrrolidin-3-ylmethyl-N-isopropyl-3-(3-methoxy-propoxy)-4-methyl-benzamide
N-((3S,4S)-4-{Cyclopropyl-(2-tetrahydro-pyran-4-yl-acetyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-3-(3-methoxy-propoxy)-4-methyl-benzamide
N-((3S,4S)-4-{((S)-2-Cyclohexyl-2-methoxy-acetyl)-cyclopropyl-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-3-(3-methoxy-propoxy)-4-methyl-benzamide
N-((3S,4S)-4-{((S)-2-Cyclohexy-2-methoxy-acetyl)-methyl-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-3-(3-methoxy-propoxy)-4-methyl-benzamide
N-((3S,4S)-4-{((S)-2-Hydroxy-3-methyl-butyryl)-methyl-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-3-(3-methoxy-propoxy)-4-methyl-benzamide
N-(3 S,4S)-4-({2-(1-Acetyl-piperidin-4-yl)-acetyl-cyclopropyl-amino}-methyl)-pyrrolidin-3-ylmethyl-N-isopropyl-3-(3-methoxy-propoxy)-4-methyl-benzamide
N-((3S,4S)-4-{((S)-2-Hydroxy-4-methyl-pentanoyl)-methyl-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-3-(3-methoxy-propoxy)-4-methyl-benzamide
N-((3S,4S)-4-((cis-4Hydroxy-cyclohexanecarbonyl)-methyl-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-3-(3-methoxy-propoxy)-4-methyl-benzamide
N-((3S,4S)-4-(((R)-3-Hydroxy-3-phenyl-propionyl)-methyl-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-3-(3-methoxy-propoxy)-4-methyl-benzamide
N-((3S,4S)-4-{((S)-3-Hydroxy-3-phenyl-propionyl)-methyl-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-3-(3-methoxy-propoxy)-4-methyl-benzamide
N-(3S,4S)-4-({2-(1-Acetyl-piperidin-4-yl)-acetyl-methyl-amino}-methyl)-pyrrolidin-3-ylmethyl-N-isopropyl-3-(3-methoxy-propoxy)-4-methyl-benzamide
N-((3S,4S)-4-{Cyclopropyl-(cis-4-hydroxy-cyclohexanecarbonyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-3-(3-methoxy-propoxy)-4-methyl-benzamide
N-((3S,4S)-4-{((S)-2-Hydroxy-3-phenyl-propionyl)-methyl-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-3-(3-methoxy-propoxy)-4-methyl-benzamide
N-((3S,4S)-4-{((2-Furan-2-yl-acetyl)-methyl-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-3-(3-methoxy-propoxy)-4-methyl-benzamide
N-((3S,4S)-4-{Cyclopropyl-((S)-2-hydroxy-4-methyl-pentanoyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-3-(3-methoxy-propoxy)-4-methyl-benzamide
Indan-2-carboxylic acid (3S,4S)-4-({isopropyl-3-(3-methoxy-propoxy)-4-methyl-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-amide
N-Isopropyl-3-(3-methoxy-propoxy)-4-methyl-N-{(3S,4S)-4-(2-methyl-2-phenyl-propionylamino)-methyl-pyrrolidin-3-ylmethyl}-benzamide
N-Isopropyl-3-(3-methoxy-propoxy)-4-methyl-N-{(3S ,4S)-4-(2-tetrahydro-pyran-4-yl-acetylamino)-methyl-pyrrolidin-3-ylmethyl}-benzamide
(S)-2,3-Dihydro-benzo1,4dioxine-2-carboxylic acid (3S,4S)-4-({isopropyl-3-(3-methoxy-propoxy)-4-methyl-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-amide
N-Isopropyl-3-(3-methoxy-propoxy)-4-methyl-N-((3S,4S)-4-{methyl-((R)-2-tetrahydro-pyran-2-yl-acetyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-benzamide
N-Isopropyl-3-(3-methoxy-propoxy)-4-methyl-N-((3S,4S)-4-{methyl-((S)-2-tetrahydro-pyran-2-yl-acetyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-benzamide
N-((3S,4S)-4-{Cyclopropyl-((R)-2-tetrahydro-furan-2-yl-acetyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-3-(3-methoxy-propoxy)-4-methyl-benzamide
N-((3S,4S)-4-{Cyclopropyl-((S)-2-tetrahydro-furan-2-yl-acetyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-N-isopropyl-3-(3-methoxy-propoxy)-4-methyl-benzamide
N-Isopropyl-N-((3S,4S)-4-{(cis-4-methoxy-cyclohexanecarbornyl)-methyl-amino-methyl}-pyrrolidin-3-ylmethyl)-3-(3-methoxy-propoxy)-4-methyl-benzamide
N-Isopropyl-N-((3S,4S)-4-{(trans-4-methoxy-cyclohexanecarbonyl)-methyl-amino-methyl}-pyrrolidin-3-ylmethyl)-3-(3-methoxy-propoxy)-4-methyl-benzamide
N-Isopropyl-N-((3S,4S)-4-{(cis-4-methoxy-cyclohexanecarbonyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-3-(3-methoxy-propoxy)-4-methyl-benzamide
N-Isopropyl-N-((3S,4S)-4-{(trans-4-methoxy-cyclohexanecarbonyl)-amino-methyl}-pyrrolidin-3-ylmethyl)-3-(3-methoxy-propoxy)-4-methyl-benzamide
1-(3-Methoxy-propyl)-1H-indole-6-carboxylic acid isopropyl-{(3S,4S)-4-(methyl-phenylacetyl-amino) -methyl-pyrrolidin-3-ylmethyl}-amide
N-Cyclopropyl-N-{(3S,4S)-4-(cyclopropyl-phenylacetyl-amino)-methyl-pyrrolidin-3-ylmethyl}-4-methoxy-3-(3-methoxy-propoxy)-benzamide
Cyclopropyl-(3S,4S)-4-({cyclopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid benzyl ester
Cyclopropyl-(3S,4S)-4-({cyclopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid isobutyl ester
Cyclopropyl-(3S,4S)-4-({cyclopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid tetrahydro-pyran-4-yl ester
Cyclopropyl-(3S*,4S*)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid benzyl ester
Cyclopropyl-(3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid benzyl ester
Cyclopropyl-(3S*,4S*)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid isobutyl ester
Cyclopropyl-(3S*,4S*)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid pyridin-4-ylmethyl ester
Cyclopropyl-(3S*,4S*)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid 1-methyl-piperidin-4-ylmethyl ester
Cyclopropyl-(3S*,4S*)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid 2-methoxy-ethyl ester
Cyclopropyl-(3S*,4S*)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid tetrahydro-pyran-4-ylmethyl ester
Cyclopropyl-(3S*,4S*)-4-({isopropyl-4-methoxy3(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid 2,2-dimethyl-propyl ester
Cyclopropyl-(3S*,4S*)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid 1-methyl-cyclopropylmethyl ester
Cyclopropyl-(3S*,4S*)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid 2-acetylamino-2-methyl-propyl ester
Cyclopropyl-(3S*,4S*)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}- methyl)-pyrrolidin-3-ylmethyl-carbamic acid phenyl ester
Cyclopropyl-(3S*,4S*)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid 2-methyl-2-methylcarbamoyl-propyl ester
Cyclopropyl-(3S*,4S*)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid 1-acetylamino-cyclopentylmethyl ester
Cyclopropyl-(3S*,4S*)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid 1-acetyl-piperidin-4-ylmethyl ester
Cyclopropyl-(3S*,4S*)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid 5-methyl-isoxazol-3-ylmethyl ester
Cyclopropyl-(3S*,4S*)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid naphthalen-1-yl ester
Cyclopropyl-(3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}methyl)-pyrrolidin-3-ylmethyl-carbamic acid cyclopropylmethyl ester
Cyclopropyl-(3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid isobutyl ester
Cyclopropyl-(3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid 4-methoxy phenyl ester
Cyclopropyl-(3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid cyclohexyl ester
Cyclopropyl-(3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid naphthalen-2-yl ester
Cyclopropyl-(3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid tetrahydro-pyran-4-yl ester
Cyclopropyl-(3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxypropoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid 5methyl-1,3dioxan-5-ylmethyl ester
Cyclopropyl-(3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxypropoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid 3(2-oxo-pyrrolidin-1-yl)-phenyl ester
Cyclopropyl-(3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid 3-morpholin-4-yl-phenyl ester
Cyclopropyl-(3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid (R)-1-(tetrahydro-furan-2-yl)methyl ester
Cyclopropyl-(3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid (R)-1-phenyl-propyl ester
Cyclopropyl-(3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid (R)-1-phenyl-ethyl ester
Cyclopropyl-(3S,4S)-4-(isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid phenyl ester
Cyclopropyl-(3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid 2-methoxy phenyl ester
Cyclopropyl-(3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid 3-methoxy-3-methyl-butyl ester
Cyclopropyl-(3S, 4S)-4-({isopropyl-4-ethoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid (R)-(tetrahydro-furan-3-yl)ester
Cyclopropyl-(3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid (S)-(tetrahydro-furan-3-yl)ester
(3S,4S)-4-({Isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-methyl-carbamic acid 3-methoxy-3-methyl-butyl ester
(3S,4S)-4-({Isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-methyl-carbamic acid tetrahydro-pyran-4-yl ester
Cyclopropyl-(3S,4S)-4-({isopropyl-3-(3-methoxy-propoxy)-4-methyl-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid tetrahydro-pyran-4-yl ester
Cyclopropyl-(3S,4S)-4-({isopropyl-3-(3-methoxy-propoxy)-4-methyl-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid (S)-(tetrahydro-furan-3-yl)ester
(3S,4S)-4-({Isopropyl-3-(3-methoxy-propoxy)-4-methyl-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-methyl-carbamic acid tetrahydro-pyran-4-yl ester
(3S,4S)-4-({Isopropyl-3-(3-methoxy-propoxy)-4-methyl-benzoyl-amino}-methyl)-pyrroidin-3- ylmethyl-methyl-carbamic acid (S)-(tetrahydro-furan-3-yl)ester
(3S,4S)-4-({Isopropyl-3-(3-methoxy-propoxy)-4-methyl-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-methyl-carbamic acid 3-methoxy-3-methyl-butyl ester
Cyclopropyl-(3S,4S)-4-({isopropyl-3-(3-methoxy-propoxy)-4-methyl-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid 3-methoxy-3-methyl-butyl ester
(3S,4S)-4-({Isopropyl-3-(3-methoxy-propoxy)-4-methyl-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-methyl-carbamic acid 4-methoxy phenyl ester
(3S,4S)-4-({Isopropyl-3-(3-methoxy-propoxy)-4-methyl-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-methyl-carbamic acid (R)-1-(tetrahydro-furan-2-yl)methyl ester
Cyclopropyl-(3S,4S)-4-({isopropyl-3-(3-methoxy-propoxy)-4-methyl-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid 4-methoxy phenyl ester
Cyclopropyl-(3S,4S)-4-({isopropyl-3-(3-methoxy-propoxy)-4-methyl-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid (R)-1-(tetrahydro-furan-2-yl)methyl ester
(3S ,4S)-4-({Isopropyl-3-(3-methoxy-propoxy)-4-methyl-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-methyl-carbamic acid 5-methyl-1,3dioxan-5-ylmethyl ester
Cyclopropyl-(3S,4S)-4-({isopropyl-3-(3-methoxy-propoxy)-4-methyl-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid 5-methyl-isoxazol-3-ylmethyl ester
(3S,4S)-4-({Isopropyl-3-(3-methoxy-propoxy)-4-methyl-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-methyl-carbamic acid 5-methyl-isoxazol-3-ylmethyl ester
Cyclopropyl-(3S,4S)-4-({4-ethyl-3-(3-methoxy-propoxy)-benzoyl-isopropyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid benzyl ester
Cyclopropyl-(3S,4S)-4-({4-ethyl-3-(3-methoxy-propoxy)-benzoyl-isopropyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid tetrahydro-pyran-4-yl ester
Cyclopropyl-(3S,4S)-4-({4-ethyl-3-(3-methoxy-propoxy)-benzoyl-isopropyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid 4methoxy phenyl ester
(3S,4S)-4-({4-Ethyl-3-(3-methoxy-propoxy)-benzoyl-isopropyl-amino}-methyl)-pyrrolidin-3-ylmethyl-methyl-carbamic acid tetrahydro-pyran-4-yl ester
(3S,4S)-4-({4-Ethyl-3-(3-methoxy-propoxy)-benzoyl-isopropyl-amino}-methyl)-pyrrolidin-3-ylmethyl-methyl-carbamic acid (R)-1-(tetrahydro-furan-2-yl)methyl ester
(3S,4S)-4-({4-Ethyl-3-(3-methoxy-propoxy)-benzoyl-isopropyl-amino}-methyl)-pyrrolidin-3-ylmethyl-methyl-carbamic acid (S)-(tetrahydro-furan-3-yl)ester
(3S,4S)-4-({4-Ethyl-3-(3-methoxy-propoxy)-benzoyl-isopropyl-amino}-methyl)-pyrrolidin-3-ylmethyl-methyl-carbamic acid 5-methyl-1,3dioxan-5-ylmethyl ester
(3S,4S)-4-({4-Ethyl-3-(3-methoxy-propoxy)benzoyl-isopropyl-amino}-methyl)-pyrrolidin-3-ylmethyl-methyl-carbamic acid 3-methoxy-3-methyl-butyl ester
Cyclopropyl-(3S,4S)-4-({isopropyl-1-(3-methoxy-propyl)-3-methyl-1H-indole-6-carbonyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid benzyl ester
Cyclopropyl-(3S,4S)-4-({isopropyl-1-(3-methoxy-propyl)-3-methyl-1H-indole-6-carbonyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid isobutyl ester
Cyclopropyl-(3S,4S)-4-({isopropyl-1-(3-methoxy-propyl)-3-methyl-1H-indole-6-carbonyl-amino}-methyl)-pyrrolidin-3-ylmethyl-carbamic acid tetrahydro-pyran-4-yl ester
Benzyl-methyl-carbamic acid (3S*,4S*)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl ester
Diisobutyl-carbamic acid (3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl ester
Benzyl-cyclopropyl-carbamic acid (3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl ester
Isobutyl-methyl-carbamic acid (3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl ester
Cyclopropyl-(tetrahydro-pyran-4-ylmethyl)-carbamic acid (3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl ester
Cyclopropyl-(tetrahydro-pyran-4-yl)-carbamic acid (3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl ester
Cyclohexylmethyl-methyl-carbamic acid (3S,4S)-4-({4-ethyl-3-(3-methoxy-propoxy)-benzoyl-isopropyl-amino}-methyl)-pyrrolidin-3-ylmethyl ester
Benzyl-cyclopropyl-carbamic acid (3S,4S)-4-({4-ethyl-3-(3-methoxy-propoxy)-benzoyl-isopropyl-amino}-methyl)-pyrrolidin-3-ylmethyl ester
Cyclopropyl-(tetrahydro-pyran-4-ylmethyl)-carbamic acid (3S,4S)-4-({4-ethyl-3-(3-methoxy-propoxy)-benzoyl-isopropyl-amino}- methyl)-pyrrolidin-3-ylmethyl ester
Cyclopropyl-(tetrahydro-pyran-3-ylmethyl)-carbamic acid (3S,4S)-4-({4-ethyl-3-(3-methoxy-propoxy)-benzoyl-isopropyl-amino}-methyl)-pyrrolidin-3-ylmethyl ester
Cyclopropyl-(tetrahydro-pyran-4-yl)-carbamic acid (3S,4S)-4-({4-ethyl-3-(3-methoxy-propoxy)-benzoyl-isopropyl-amino}-methyl)-pyrrolidin-3-ylmethyl ester
Cyclopropyl-(tetrahydro-pyran-2-ylmethyl)-carbamic acid (3S,4S)-4-({4-ethyl-3-(3-methoxy-propoxy)-benzoyl-isopropyl-amino}-methyl)-pyrrolidin-3-ylmethyl ester
Cyclopropyl-(tetrahydro-pyran-4-yl)-carbamic acid (3S,4S)-4-({isopropyl-1-(3-methoxy-propyl)-3-methyl-1H-indole-6-carbonyl-amino}-methyl)-pyrrolidin-3-ylmethyl ester
((R)-1-Phenyl-propyl)-carbamic acid (3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl ester
N-(3S*,4S*)-4-(1-Cyclopropyl-3-furan-2-ylmethyl-ureidomethyl)-pyrrolidin-3-ylmethyl-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-(3S,4S)-4-(1-Cyclopropyl-3-furan-2-ylmethyl-ureidomethyl)-pyrrolidin-3-ylmethyl-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-(3S*,4S*)-4-(3-(4-Methoxy benzyl-1-cyclopropyl-ureidomethyl)-pyrrolidin-3-ylmethyl-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-(3S*,4S*)-4-(3-(4-Chloro benzyl-1-cyclopropyl-ureidomethyl)-pyrrolidin-3-ylmethyl-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N(3S*,4S*)-4-(3-(4-Fluoro benzo-1-cyclopropyl-ureidomethyl)-pyrrolidin-3-ylmethyl-N-isopropyl-4 -methoxy-3-(3-methoxy-propoxy)-benzamide
N-(3S*,4S*)-4-(3-Cyclohexylmethyl-1-cyclopropyl-ureidomethyl)-pyrrolidin-3-ylmethyl-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-{(3S*,4S*)-4-1-Cyclopropyl-3-(tetrahydro-pyran-4-ylmethyl)-ureidomethyl-pyrolidin-3-ylmethyl}-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-(3S*,4S*)-4-(1-Cyclopropyl-3-phenethyl-ureidomethyl)-pyrrolidin-3-ylmethyl-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-(3S*,4S*)-4-(1-Cyclopropyl-3,3-diphenyl-ureidomethyl)-pyrrolidin-3-ylmethyl-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-(3S*,4S*)-4-(1-Cyclopropyl-3,3-diisopropyl-ureidomethyl)-pyrrolidin-3-ylmethyl-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-(3S*,4S*)-4-(3-Benzyl-1-cyclopropyl-3-methyl-ureidomethyl)-pyrrolidin-3-ylmethyl-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-(3S*,4S*)-4-(3-Benzyl-1-cyclopropyl-3-ethyl-ureidomethyl)-pyrrolidin-3-ylmethyl-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-(3S,4S)-4-(3-Benzyl-1-cyclopropyl-3-ethyl-ureidomethyl)-pyrrolidin-3-ylmethyl-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-(3S*,4S*)-4-(3-Benzyl-1,3-dicyclopropyl-ureidomethyl)-pyrrolidin-3-ylmethyl-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-(3S*,4S*)-4-(1-Cyclopropyl-3-phenyl-ureidomethyl)-pyrrolidin-3-ylmethyl-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-(3S*,4S*)-4-3-Benzhydryl-1-cyclopropyl-ureidomethyl)-pyrrolidin-3-ylmethyl-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-(3S,4S)-4-(3-Benzyl-1-cyclopropyl-ureidomethyl)-pyrrolidin-3-ylmethyl-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-(3S,4S)-4-(1,3-Dicyclopropyl-3-phenyl-ureidomethyl)-pyrrolidin-3-ylmethyl-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-(3S,4S)-4(3-Cyclohexyl-1-cyclopropyl-ureidomethyl)-pyrrolidin-3-ylmethyl-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-(3S*,4S*)-4-(1-Cyclopropyl-3-naphthalen-1-yl-ureidomethyl)-pyrrolidin-3-ylmethyl-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-(3S,4S)-4-(1-Cyclopropyl-3-naphthalen-2-ylureidomethyl)-pyrrolidin-3-ylmethyl-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-{(3S,4S)-4-1-Cyclopropyl-3-((R)-1-phenyl-propyl)-ureidomethyl-pyrrolidin-3-ylmethyl}-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-(3S,4S)-4-(1-Cyclopropyl-3-isobutyl-3-methyl-ureidomethyl)-pyrrolidin-3-ylmethyl-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
N-{(3S,4S)-4-1-Cyclopropyl-3-((S)-1-phenyl-propyl)-ureidomethyl-pyrrolidin-3-ylmethyl}-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
(R)-3-Phenyl-pyrrolidine-1-carboxylic acid cyclopropyl-(3S,4S)-4-({isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-amide
4-Ethyl-3-(3-hydroxy-propoxy)-N-isopropyl-N-{(3S,4S)-4-(methyl-phenylacetyl-amino)-methyl-pyrrolidin-3-ylmethyl}-benzamide
N-{(3S,4S)-4-(Cyclopropyl-phenylacetyl-amino)-methyl-pyrrolidin-3-ylmethyl}-3-(3-hydroxy-propoxy)-N-isopropyl-4-methoxy-benzamide
N-{(3S*,4S*)-4-(Cyclopropyl-phenylacetyl-amino)-methyl-pyrrolidin-3-ylmethyl}-N-isopropyl-4-methoxy-3-(4-methoxy-butyl)-benzamide
N-{(3S*,4S*)-4-(Cyclopropyl-phenylacetyl-amino)-methyl-pyrrolidin-3-ylmethyl}-4-difluoromethyl-N-isopropyl-3-(3-methoxy-propoxy)-benzamide
8-(3-Methoxy-propoxy)-2,3-dihydro-benzo1,4dioxine-6-carboxylic acid {(3S*,4S*)-4-(cyclopropyl-phenylacetyl-amino)-methyl-pyrrolidin-3-ylmethyl}-isopropyl-amide
N-{(3S*,4S*)-4-(Cyclopropyl-phenylacetyl-amino)-methyl-pyrrolidin-3-ylmethyl}-N-isopropyl-4-methoxy-5-(3-methoxy-propoxy)-2-methyl-benzamide
2-Chloro-N-{(3S*,4S*)-4-(cyclopropyl-phenylacetyl-amino)methyl-pyrrolidin-3-ylmethyl}-N-isopropyl-4-methoxy-5-(3-methoxy-propoxy)-benzamide
3-Chloro-N-{(3S*,4S*)-4-(cyclopropyl-phenylacetyl-amino)-methyl-pyrrolidin-3-ylmethyl}-N-isopropyl-5-(3-methoxy-propoxy)-benzamide
4-Chloro-N-{(3S*4S*)-4-(cyclopropyl-phenylacetyl-amino)-methyl-pyrrolidin-3-ylmethyl}-N-isopropyl-3-(3-methoxy-propoxy)-benzamide
4-tert-Butyl-N-isopropyl-3-(3-methoxy-propoxy)-N-{(3S,4S)-4-(methyl-phenylacetyl-amino)-methyl-pyrrolidin-3-ylmethyl}-benzamide
N-Isopropyl-4-methoxy-3-(2-methoxy-ethoxymethyl)-N-{(3S,4S)-4-(methyl-phenylacetyl-amino)-methyl-pyrrolidin-3-ylmethyl}-benzamide
N-Isopropyl-3-(2-methoxy-ethoxymethyl)-N-{(3S,4S)-4-(methyl-phenylacetyl-amino)-methyl-pyrrolidin-3-ylmethyl}-4-trifluoromethoxy-benzamide
N-Isopropyl-4-methoxy-N-{(3S,4S)-4-(methyl-phenylacetyl-amino)-methyl-pyrrolidin-3-ylmethyl}-3-(3,3,3-trifluoro-propoxy)-benzamide
N-Isopropyl-4-methoxy-N-{(3S,4S)-4(methyl-phenylacetyl-amino)-methyl-pyrrolidin-3-ylmethyl}-3-(4,4,4-trifluoro-butoxy)-benzamide
N-{(3S,4S)-4-(Cyclopropyl-phenylacetyl-amino)-methyl-pyrrolidin-3-ylmethyl}-N-isopropyl-4-methoxy-3-(3-trifluoromethoxy-propoxy)-benzamide
N-{(3S,4S)-4-(Cyclopropyl-phenylacetyl-amino)-methyl-pyrrolidin-3-ylmethyl}-4-ethyl-N-isopropyl-3-(3-trifluoromethoxy-propoxy)-benzamide
N-Isopropyl-4-methoxy-3-(5-methyl-isoxazol-3-ylmethoxy)-N-{(3S,4S)-4-(methyl-phenylacetyl-amino)-methyl-pyrrolidin-3-ylmethyl}-benzamide
N-{(3S,4S)-4-(Cyclopropyl-phenylacetyl-amino)-methyl-pyrrolidin-3-ylmethyl}-N-isopropyl-3-(2-methoxy-ethoxymethyl)-4-trifluoromethoxy-benzamide
3-(2-Ethoxy-ethoxy)-N-isopropyl-4-methoxy-N-{(3S,4S)-4-(methyl-phenyl acetyl-amino)-methyl-pyrrolidin-3-ylmethyl}-benzamide
N-(3S*,4S*)-4-({Cyclopropyl-2-(4-methoxy-phenyl)-acetyl-amino}-methyl)-pyrrolidin-3-ylmethyl-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide and
N-(3S*,4S*)-4-({Cyclopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzoyl-amino}-methyl)-pyrrolidin-3-ylmethyl-N-isopropyl-4-methoxy-3-(3-methoxy-propoxy)-benzamide
or a pharmaceutically acceptable salt thereof.
5. The compound according to claim 1 with the formula
or a pharmaceutically acceptable salt thereof.
6. A pharmaceutical composition, comprising:
a compound of the formula I according to claim 1, or a pharmaceutically acceptable salt thereof and
a pharmaceutically acceptable carrier material.
7. A method of treating hypertension, comprising:
administering to a warm-blooded animal in need of such treatment a pharmaceutically effective amount of a compound of the formula I according to claim 1, or a pharmaceutically acceptable salt thereof.